Dosing & Administration
Adult Dose
Start 3.125 mg PO BID, target 25 mg BID (take with food).
Pediatric Dose
0.1 mg/kg/dose PO BID.
Renal Adjustment
No adjustment necessary.
Hepatic Adjustment
Contraindicated in severe impairment.
Safety & Special Populations
Pregnancy Category
C
Lactation Safety
Unknown, avoid if possible.
Contraindications & Adverse Effects
Contraindications
- Severe bradycardia
- Asthma/Severe COPD
- Decompensated HF
Common Adverse Effects
- Hypotension
- Fatigue
- Bradycardia
- Weight gain