Sumatriptan (Imitrex)

Neurology (5-HT1 Agonist / Triptan)

Dosing & Administration

Adult Dose

50-100 mg PO (repeat once after 2h if needed, max 200 mg/day). SQ: 6 mg (max 12 mg/day).

Pediatric Dose

Not FDA approved < 18 yrs, but sometimes used off-label.

Renal Adjustment

No adjustment necessary.

Hepatic Adjustment

Max 50 mg PO single dose in mild-mod impairment.

Safety & Special Populations

Pregnancy Category

C

Lactation Safety

Compatible (discard milk for 8h optionally to minimize exposure).

Contraindications & Adverse Effects

Contraindications

  • Ischemic heart disease
  • Prinzmetal angina
  • Uncontrolled hypertension
  • History of stroke

Common Adverse Effects

  • Chest tightness / pressure
  • Flushing
  • Tingling