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Drug Dilution Guide

Standard concentrations, recommended diluents, and administration rates for common IV medications.

Norepinephrine

Standard Diluent

D5W or NS

Final Concentration

4 mg / 250 mL (16 mcg/mL) or 8 mg / 250 mL (32 mcg/mL)

Infusion Rate

Titrate to MAP > 65 mmHg (usually 1 - 30 mcg/min)

Max: No absolute max, but > 30 mcg/min implies profound shock

Stability

24 hours at room temp

Administration Notes

Central line preferred due to extravasation risk. D5W is traditionally preferred to prevent oxidation, though NS is commonly used.

Amiodarone

Standard Diluent

D5W

Final Concentration

900 mg / 500 mL (1.8 mg/mL)

Infusion Rate

1 mg/min for 6 hrs, then 0.5 mg/min for 18 hrs

Stability

24 hours

Administration Notes

Requires in-line filter. Use glass or polyolefin bags to prevent PVC adsorption.

Insulin (Regular)

Standard Diluent

Normal Saline (0.9% NaCl)

Final Concentration

100 Units / 100 mL (1 Unit/mL)

Infusion Rate

0.1 Units/kg/hr (DKA/HHS protocol)

Stability

24 hours

Administration Notes

Flush tubing with 20-50 mL of solution before connecting to patient due to insulin binding to plastic tubing.

Epinephrine

Standard Diluent

D5W or NS

Final Concentration

4 mg / 250 mL (16 mcg/mL)

Infusion Rate

Titrate to effect (usually 1 - 10 mcg/min)

Max: No absolute max; depends on clinical response

Stability

24 hours at room temp

Administration Notes

Central line strongly preferred. Can cause profound tachycardia and ischemia.

Vasopressin

Standard Diluent

D5W or NS

Final Concentration

40 Units / 100 mL (0.4 Units/mL)

Infusion Rate

0.03 - 0.04 Units/min (septic shock)

Max: 0.04 Units/min (higher doses risk splanchnic ischemia)

Stability

24 hours

Administration Notes

Not titrated like other pressors; usually set at a fixed rate as an adjunct to Norepinephrine.

Propofol

Standard Diluent

Ready to use (lipid emulsion)

Final Concentration

10 mg/mL

Infusion Rate

5 - 50 mcg/kg/min

Max: Generally avoid > 80 mcg/kg/min for prolonged periods

Stability

12 hours (due to lipid emulsion infection risk)

Administration Notes

Strict aseptic technique required. Monitor triglycerides if infused > 48 hours to avoid PRIS.

Dexmedetomidine

Standard Diluent

NS

Final Concentration

400 mcg / 100 mL (4 mcg/mL)

Infusion Rate

0.2 - 1.5 mcg/kg/hr

Max: 1.5 mcg/kg/hr

Stability

24 hours

Administration Notes

Does not cause respiratory depression. Watch for bradycardia and hypotension.

Fentanyl

Standard Diluent

NS or D5W

Final Concentration

1,000 mcg / 100 mL (10 mcg/mL) or 2,500 mcg / 250 mL

Infusion Rate

25 - 200 mcg/hr

Max: Titrate to RASS/pain scores

Stability

24 hours

Administration Notes

Highly lipophilic, accumulates in fat with prolonged infusions.

Heparin

Standard Diluent

D5W or NS

Final Concentration

25,000 Units / 250 mL (100 Units/mL)

Infusion Rate

Weight-based protocol (e.g., 12-18 Units/kg/hr)

Max: Per nomogram

Stability

24 hours

Administration Notes

Monitor aPTT or Anti-Xa levels strictly. Watch for HIT (platelet drop).

Nitroglycerin

Standard Diluent

D5W or NS

Final Concentration

50 mg / 250 mL (200 mcg/mL)

Infusion Rate

5 - 200 mcg/min

Max: 200 mcg/min

Stability

24 hours

Administration Notes

Requires glass bottles or special non-PVC tubing to prevent adsorption.

Diltiazem

Standard Diluent

NS or D5W

Final Concentration

125 mg / 125 mL (1 mg/mL)

Infusion Rate

5 - 15 mg/hr

Max: 15 mg/hr

Stability

24 hours

Administration Notes

Usually preceded by a 0.25 mg/kg bolus over 2 minutes.

Dobutamine

Standard Diluent

D5W or NS

Final Concentration

500 mg / 250 mL (2,000 mcg/mL)

Infusion Rate

2 - 20 mcg/kg/min

Max: 20 mcg/kg/min

Stability

24 hours

Administration Notes

Inotrope. May cause significant tachycardia and arrhythmias. Can cause hypotension if patient is volume depleted.

Milrinone

Standard Diluent

D5W or NS

Final Concentration

20 mg / 100 mL (200 mcg/mL)

Infusion Rate

0.375 - 0.75 mcg/kg/min

Max: 0.75 mcg/kg/min

Stability

72 hours

Administration Notes

Inodilator. Needs renal dose adjustment. May drop blood pressure significantly.

Nicardipine

Standard Diluent

NS or D5W

Final Concentration

25 mg / 250 mL (0.1 mg/mL)

Infusion Rate

5 - 15 mg/hr

Max: 15 mg/hr

Stability

24 hours

Administration Notes

Change site every 12 hours if peripheral to avoid phlebitis. Central line preferred.

Labetalol

Standard Diluent

D5W

Final Concentration

200 mg / 200 mL (1 mg/mL)

Infusion Rate

2 - 8 mg/min

Max: 8 mg/min (Total max 300mg in 24 hours)

Stability

24 hours

Administration Notes

Avoid in patients with severe asthma or bradycardia (non-selective beta blocker).

Phenylephrine

Standard Diluent

NS or D5W

Final Concentration

40 mg / 250 mL (160 mcg/mL) or 100 mg / 250 mL (400 mcg/mL)

Infusion Rate

10 - 200 mcg/min

Max: 200 mcg/min

Stability

24 hours

Administration Notes

Pure alpha-1 agonist. Can cause reflex bradycardia.

Ketamine

Standard Diluent

NS or D5W

Final Concentration

500 mg / 50 mL (10 mg/mL)

Infusion Rate

1 - 10 mcg/kg/min (Analgesia/Sedation)

Max: Depends on indication

Stability

24 hours

Administration Notes

Does not usually drop blood pressure; may actually increase sympathetic tone. Can cause emergence delirium.

Cisatracurium

Standard Diluent

D5W or NS

Final Concentration

100 mg / 50 mL (2 mg/mL) or 200 mg / 100 mL

Infusion Rate

1 - 3 mcg/kg/min

Max: Titrate to Train of Four (TOF) usually 1-2 twitches

Stability

24 hours refrigerated, shorter at room temp

Administration Notes

Requires secure airway and mechanical ventilation. Independent of hepatic/renal function (Hoffmann elimination).

Pantoprazole

Standard Diluent

NS

Final Concentration

80 mg / 100 mL (0.8 mg/mL)

Infusion Rate

8 mg/hr

Max: 8 mg/hr

Stability

12 hours (protect from light if prolonged)

Administration Notes

Use dedicated line or flush thoroughly. Incompatible with many drugs.

Octreotide

Standard Diluent

NS

Final Concentration

500 mcg / 500 mL (1 mcg/mL)

Infusion Rate

25 - 50 mcg/hr

Max: 50 mcg/hr

Stability

24 hours

Administration Notes

Used for esophageal variceal bleeding. Often started with a 50 mcg IV push bolus.

Magnesium Sulfate

Standard Diluent

NS or D5W

Final Concentration

4 g / 100 mL or 4 g / 250 mL

Infusion Rate

1 - 2 g/hr (replacement) or 2 g over 10 min (Torsades)

Max: Varies; high rates used for eclampsia/Torsades

Stability

24 hours

Administration Notes

Monitor deep tendon reflexes and respiratory rate if using high doses.

Adenosine

Standard Diluent

Undiluted (Rapid IV Push)

Final Concentration

3 mg/mL

Infusion Rate

6 mg rapid IV push, followed by 12 mg if needed

Max: Give over 1-2 seconds

Stability

Room temperature

Administration Notes

Requires immediate rapid 20 mL NS flush and elevation of the extremity. Half-life is < 10 seconds.

Alteplase (tPA)

Standard Diluent

Sterile Water

Final Concentration

1 mg/mL

Infusion Rate

Stroke: 0.9 mg/kg (10% as bolus, 90% over 1 hour)

Max: Max total dose 90 mg (for stroke)

Stability

Use within 8 hours of reconstitution

Administration Notes

Strict BP control required (< 185/110) before and during administration.

Aminophylline

Standard Diluent

D5W or NS

Final Concentration

1 mg/mL or 2 mg/mL

Infusion Rate

0.5 - 0.7 mg/kg/hr

Max: Depends on serum theophylline levels

Stability

24 hours

Administration Notes

Narrow therapeutic index. Monitor for arrhythmias and seizures.

Atracurium

Standard Diluent

NS or D5W

Final Concentration

0.2 mg/mL or 0.5 mg/mL

Infusion Rate

5 - 10 mcg/kg/min

Max: Titrate to TOF

Stability

Refrigerate intact vials; degrades rapidly at room temp

Administration Notes

Can cause histamine release (hypotension, tachycardia).

Atropine

Standard Diluent

Undiluted

Final Concentration

0.1 mg/mL or 1 mg/mL

Infusion Rate

1 mg IV push every 3-5 mins (Bradycardia)

Max: Max total dose 3 mg

Stability

Room temperature

Administration Notes

Paradoxical bradycardia can occur with doses < 0.5 mg or slow administration.

Bivalirudin

Standard Diluent

D5W or NS

Final Concentration

5 mg/mL

Infusion Rate

0.15 - 0.2 mg/kg/hr (titrated to aPTT)

Max: Per nomogram

Stability

24 hours

Administration Notes

Direct thrombin inhibitor. Preferred in patients with HIT history.

Bumetanide

Standard Diluent

D5W or NS

Final Concentration

0.25 mg/mL

Infusion Rate

0.5 - 2 mg/hr (continuous infusion)

Max: Max 10 mg/day

Stability

24 hours

Administration Notes

Loop diuretic. ~40x more potent than furosemide (1 mg bumetanide = 40 mg furosemide).

Caspofungin

Standard Diluent

NS (Do NOT use Dextrose)

Final Concentration

0.5 mg/mL

Infusion Rate

Infuse over 1 hour

Max: Avoid rapid infusion (histamine release)

Stability

24 hours (Room Temp) or 48 hours (Refrigerated)

Administration Notes

Echinocandin antifungal. Specifically incompatible with dextrose-containing solutions.

Cefepime

Standard Diluent

NS or D5W

Final Concentration

10 - 40 mg/mL

Infusion Rate

Give over 30 mins (Standard) or 3-4 hours (Extended Infusion)

Max: Avoid rapid push

Stability

24 hours (Room Temp)

Administration Notes

Neurotoxicity (encephalopathy, seizures) risk in renal failure if not dose adjusted.

Dexamethasone

Standard Diluent

Undiluted (IV Push) or 50mL NS/D5W

Final Concentration

4 mg/mL or 10 mg/mL

Infusion Rate

Push over 1-2 mins or infuse over 15 mins

Max: Varies by indication

Stability

24 hours

Administration Notes

Rapid IV push can cause intense perineal burning sensation.

Digoxin

Standard Diluent

NS, D5W, or Undiluted

Final Concentration

100 - 250 mcg/mL

Infusion Rate

Give over at least 5 minutes

Max: Avoid rapid push (vasoconstriction)

Stability

24 hours

Administration Notes

Monitor potassium closely (hypokalemia increases risk of digoxin toxicity).

Enalaprilat

Standard Diluent

Undiluted or 50mL NS/D5W

Final Concentration

1.25 mg/mL

Infusion Rate

1.25 mg IV push over 5 minutes

Max: Max 5 mg/dose every 6 hours

Stability

24 hours

Administration Notes

IV ACE inhibitor. Can cause profound, unpredictable hypotension.

Eptifibatide

Standard Diluent

NS or D5W

Final Concentration

2 mg/mL or 0.75 mg/mL

Infusion Rate

2 mcg/kg/min (ACS)

Max: 2 mcg/kg/min

Stability

Protect from light until administration

Administration Notes

Glycoprotein IIb/IIIa inhibitor. Requires renal adjustment (CrCl < 50 mL/min = 1 mcg/kg/min).

Flumazenil

Standard Diluent

Undiluted

Final Concentration

0.1 mg/mL

Infusion Rate

0.2 mg over 15 seconds (repeat up to 3 mg)

Max: 0.2 mg/min

Stability

24 hours

Administration Notes

Benzodiazepine reversal. High risk of inducing seizures in chronic benzo users.

Furosemide

Standard Diluent

Undiluted or NS/D5W

Final Concentration

10 mg/mL

Infusion Rate

Push: max 20 mg/min. Infusion: max 4 mg/min.

Max: 4 mg/min (to avoid ototoxicity)

Stability

24 hours (protect from light)

Administration Notes

Rapid push of large doses (>120mg) can cause permanent deafness.

Glucagon

Standard Diluent

Manufacturer's Diluent or Sterile Water

Final Concentration

1 mg/mL

Infusion Rate

1-5 mg IV push (Beta-blocker/CCB overdose)

Max: Infusions at 1-5 mg/hr if response to bolus

Stability

Use immediately after reconstitution

Administration Notes

Can cause severe nausea and vomiting; pretreat with antiemetics.

Haloperidol

Standard Diluent

D5W (preferred) or NS

Final Concentration

5 mg/mL

Infusion Rate

IV push over 1 min, or continuous infusion 3-25 mg/hr

Max: Depends on agitation severity

Stability

24 hours

Administration Notes

High risk of QTc prolongation and Torsades de Pointes. Baseline ECG required.

Hydralazine

Standard Diluent

Undiluted

Final Concentration

20 mg/mL

Infusion Rate

10 - 20 mg IV push over 1 minute

Max: Max 20 mg per dose

Stability

Use immediately; degrades upon contact with metal/light

Administration Notes

Onset is delayed (10-30 mins). Do not stack doses too quickly.

Hydrocortisone

Standard Diluent

NS or D5W

Final Concentration

1 mg/mL or 2 mg/mL

Infusion Rate

50-100 mg IV push, or 200 mg/24hr continuous

Max: Administer push over 3-5 mins

Stability

24 hours

Administration Notes

Drug of choice for relative adrenal insufficiency in septic shock.

Isoproterenol

Standard Diluent

D5W

Final Concentration

1 mg / 250 mL (4 mcg/mL)

Infusion Rate

2 - 10 mcg/min

Max: Titrate to heart rate

Stability

24 hours (protect from light)

Administration Notes

Pure beta agonist. Used for refractory bradycardia/heart block. Causes profound vasodilation.

Vancomycin

Standard Diluent

NS or D5W

Final Concentration

5 mg/mL

Infusion Rate

1-2 hours depending on dose

Max: 10 mg/min (to prevent Red Man Syndrome)

Stability

14 days refrigerated

Administration Notes

Requires therapeutic drug monitoring (troughs).

Meropenem

Standard Diluent

NS

Final Concentration

1 - 20 mg/mL

Infusion Rate

15-30 mins or 3-hour extended infusion

Max: 3-hour extended

Stability

24 hours refrigerated

Administration Notes

Broad spectrum carbapenem. May lower seizure threshold.

Piperacillin/Tazobactam

Standard Diluent

NS or D5W

Final Concentration

200 mg/mL

Infusion Rate

30 mins or 4-hour extended infusion

Max: 4-hour extended

Stability

24 hours room temp

Administration Notes

Extended infusion optimizes time above MIC for pseudomonas.

Linezolid

Standard Diluent

Ready to use bags (D5W)

Final Concentration

2 mg/mL

Infusion Rate

30 - 120 mins

Max: 120 mins

Stability

Room temp (protect from light)

Administration Notes

Weak MAOI; risk of serotonin syndrome with SSRIs.

Fluconazole

Standard Diluent

Ready to use (NS)

Final Concentration

2 mg/mL

Infusion Rate

1 - 2 hours

Max: 200 mg/hr

Stability

Room temp

Administration Notes

No renal adjustment for single doses.

Amphotericin B

Standard Diluent

D5W ONLY

Final Concentration

0.1 mg/mL

Infusion Rate

2 - 6 hours

Max: Over 6 hours

Stability

24 hours (protect from light)

Administration Notes

Pre-medicate with APAP/Diphenhydramine to prevent rigors.

Acyclovir

Standard Diluent

NS or D5W

Final Concentration

7 mg/mL

Infusion Rate

1 hour

Max: 1 hour minimum

Stability

24 hours room temp (do not refrigerate)

Administration Notes

Ensure adequate hydration to prevent crystal nephropathy.

Metronidazole

Standard Diluent

Ready to use (NS)

Final Concentration

5 mg/mL

Infusion Rate

30 - 60 mins

Max: 60 mins

Stability

Room temp (do not refrigerate)

Administration Notes

Disulfiram-like reaction with alcohol.

Levofloxacin

Standard Diluent

Ready to use (D5W)

Final Concentration

5 mg/mL

Infusion Rate

60 - 90 mins

Max: 90 mins

Stability

Room temp

Administration Notes

QTc prolongation risk. Adjust in renal failure.

Ciprofloxacin

Standard Diluent

Ready to use (D5W)

Final Concentration

2 mg/mL

Infusion Rate

60 mins

Max: 60 mins

Stability

Room temp

Administration Notes

Tendon rupture risk (Black Box Warning).

Azithromycin

Standard Diluent

NS or D5W

Final Concentration

1 - 2 mg/mL

Infusion Rate

1 hour (500mg) or 3 hours

Max: 1 hour minimum

Stability

24 hours

Administration Notes

Do not give as a bolus.

Ceftriaxone

Standard Diluent

NS or D5W

Final Concentration

10 - 40 mg/mL

Infusion Rate

30 mins

Max: 30 mins

Stability

3 days room temp

Administration Notes

Do not mix with calcium (e.g., Lactated Ringers).

Cefazolin

Standard Diluent

NS or D5W

Final Concentration

10 - 20 mg/mL

Infusion Rate

30 mins

Max: 30 mins

Stability

24 hours room temp

Administration Notes

Common surgical prophylaxis.

Gentamicin

Standard Diluent

NS or D5W

Final Concentration

1 - 10 mg/mL

Infusion Rate

30 - 60 mins

Max: 60 mins

Stability

24 hours

Administration Notes

Nephrotoxic and ototoxic. Requires peak/trough monitoring.

Tobramycin

Standard Diluent

NS or D5W

Final Concentration

1 - 10 mg/mL

Infusion Rate

30 - 60 mins

Max: 60 mins

Stability

24 hours

Administration Notes

Similar to gentamicin; preferred for Pseudomonas.

Esmolol

Standard Diluent

NS or D5W

Final Concentration

10 mg/mL

Infusion Rate

50 - 300 mcg/kg/min

Max: 300 mcg/kg/min

Stability

24 hours

Administration Notes

Ultra-short acting beta blocker (half-life 9 mins).

Nitroprusside

Standard Diluent

D5W ONLY

Final Concentration

200 mcg/mL

Infusion Rate

0.3 - 10 mcg/kg/min

Max: 10 mcg/kg/min (for max 10 mins)

Stability

24 hours (wrap in foil to protect from light)

Administration Notes

Risk of cyanide/thiocyanate toxicity with prolonged use.

Procainamide

Standard Diluent

NS or D5W

Final Concentration

2 - 4 mg/mL

Infusion Rate

20 - 50 mg/min (loading) then 1-4 mg/min

Max: 50 mg/min

Stability

24 hours

Administration Notes

Stop if QRS widens >50% or hypotension occurs.

Lidocaine

Standard Diluent

D5W

Final Concentration

4 mg/mL or 8 mg/mL

Infusion Rate

1 - 4 mg/min

Max: 4 mg/min

Stability

24 hours

Administration Notes

Signs of toxicity: numbness, confusion, seizures.

Epoprostenol

Standard Diluent

Special diluent

Final Concentration

3000 - 15000 ng/mL

Infusion Rate

Titrated in ng/kg/min

Max: Varies

Stability

24-48 hrs with ice packs depending on brand

Administration Notes

Pulmonary hypertension. Abrupt stopping causes rebound fatal PH crisis.

Treprostinil

Standard Diluent

NS or D5W

Final Concentration

Varies

Infusion Rate

Titrated in ng/kg/min

Max: Varies

Stability

48 hours at room temp

Administration Notes

Longer half-life than epoprostenol.

Nesiritide

Standard Diluent

D5W or NS

Final Concentration

5 mcg/mL

Infusion Rate

0.01 mcg/kg/min

Max: 0.03 mcg/kg/min

Stability

24 hours

Administration Notes

BNP analog. Used for decompensated heart failure.

Clonidine

Standard Diluent

NS

Final Concentration

15 - 30 mcg/mL

Infusion Rate

15 - 150 mcg/hr (if used IV)

Max: 150 mcg/hr

Stability

24 hours

Administration Notes

Central alpha-2 agonist. Rebound hypertension if stopped abruptly.

Phentolamine

Standard Diluent

NS

Final Concentration

1 mg/mL

Infusion Rate

Extravasation: 5-10 mg injected locally

Max: N/A

Stability

Use immediately

Administration Notes

Antidote for vasopressor extravasation.

Argatroban

Standard Diluent

NS or D5W

Final Concentration

1 mg/mL

Infusion Rate

2 mcg/kg/min

Max: 10 mcg/kg/min

Stability

24 hours

Administration Notes

Direct thrombin inhibitor. Falsely elevates INR.

Phenobarbital

Standard Diluent

NS or D5W (slow push preferred)

Final Concentration

130 mg/mL

Infusion Rate

60 mg/min (adults)

Max: 60 mg/min

Stability

Room temp

Administration Notes

Long acting barbiturate. Respiratory depression risk.

Pentobarbital

Standard Diluent

Undiluted

Final Concentration

50 mg/mL

Infusion Rate

1 - 5 mg/kg/hr

Max: Titrate to burst suppression

Stability

Use fresh

Administration Notes

Used for refractory status epilepticus or high ICP.

Thiopental

Standard Diluent

NS or Sterile Water

Final Concentration

25 mg/mL (2.5%)

Infusion Rate

Rapid IV push for induction

Max: N/A

Stability

24 hours refrigerated

Administration Notes

Highly alkaline. Causes tissue necrosis if extravasated.

Midazolam

Standard Diluent

D5W or NS

Final Concentration

1 mg/mL or 5 mg/mL

Infusion Rate

1 - 10 mg/hr (continuous)

Max: Titrate to RASS

Stability

24 hours

Administration Notes

Accumulates in renal failure (active metabolite).

Lorazepam

Standard Diluent

D5W or NS

Final Concentration

0.1 - 1 mg/mL

Infusion Rate

1 - 10 mg/hr

Max: Max 10 mg/hr

Stability

24 hours

Administration Notes

Risk of propylene glycol toxicity at high doses.

Diazepam

Standard Diluent

Undiluted (do not mix in bags)

Final Concentration

5 mg/mL

Infusion Rate

5 mg/min (push)

Max: 5 mg/min

Stability

Immediate use

Administration Notes

Binds to plastic bags/tubing. Give via slow IV push.

Remifentanil

Standard Diluent

NS or D5W

Final Concentration

50 mcg/mL

Infusion Rate

0.05 - 0.25 mcg/kg/min

Max: Varies by setting

Stability

24 hours

Administration Notes

Ultra-short acting (hydrolyzed by plasma esterases). Does not accumulate.

Sufentanil

Standard Diluent

NS or D5W

Final Concentration

5 mcg/mL

Infusion Rate

0.1 - 0.5 mcg/kg/hr

Max: Varies

Stability

24 hours

Administration Notes

5-10x more potent than fentanyl.

Morphine

Standard Diluent

NS or D5W

Final Concentration

1 mg/mL

Infusion Rate

1 - 10 mg/hr

Max: Titrate to effect

Stability

24 hours

Administration Notes

Histamine release can cause hypotension and pruritus.

Hydromorphone

Standard Diluent

NS or D5W

Final Concentration

0.2 mg/mL

Infusion Rate

0.2 - 3 mg/hr

Max: Titrate to effect

Stability

24 hours

Administration Notes

5-7x more potent than morphine.

Methadone

Standard Diluent

NS

Final Concentration

1 - 5 mg/mL

Infusion Rate

IV push

Max: N/A

Stability

Use immediately

Administration Notes

Prolongs QTc. Has NMDA antagonist properties.

Ketorolac

Standard Diluent

Undiluted

Final Concentration

15 - 30 mg/mL

Infusion Rate

IV push over 15 seconds

Max: 15 seconds

Stability

Room temp

Administration Notes

NSAID. Max duration of therapy is 5 days (GI bleed/renal risk).

Metoclopramide

Standard Diluent

NS or D5W

Final Concentration

5 mg/mL

Infusion Rate

Push over 1-2 mins

Max: 2 mins

Stability

24 hours (protect from light)

Administration Notes

Risk of EPS and tardive dyskinesia.

Ondansetron

Standard Diluent

NS or D5W

Final Concentration

2 mg/mL

Infusion Rate

Push over 2-5 mins

Max: 5 mins

Stability

24 hours

Administration Notes

QTc prolongation risk.

Promethazine

Standard Diluent

NS

Final Concentration

Max 25 mg/mL

Infusion Rate

Dilute in 50mL and give over 10-15 mins

Max: Do not give rapid push

Stability

Use immediately

Administration Notes

High risk of tissue necrosis. Dilution strongly recommended.

Erythromycin

Standard Diluent

NS

Final Concentration

1 - 5 mg/mL

Infusion Rate

3 mg/kg over 45 mins (for gastroparesis)

Max: 45 mins

Stability

8 hours at room temp

Administration Notes

Potent CYP3A4 inhibitor and QTc prolonger.

Levothyroxine

Standard Diluent

NS

Final Concentration

20 - 40 mcg/mL

Infusion Rate

IV push over 1-2 minutes

Max: 2 mins

Stability

Reconstitute immediately before use

Administration Notes

IV dose is ~50% of the oral dose.

Methylprednisolone

Standard Diluent

NS or D5W

Final Concentration

Varies

Infusion Rate

Push over 3-15 mins depending on dose

Max: High doses (>250mg) must be given over >30 mins

Stability

24 hours

Administration Notes

Used for acute spinal cord injury, MS exacerbations, COPD.

Terlipressin

Standard Diluent

NS

Final Concentration

1 mg/10 mL

Infusion Rate

1-2 mg IV push over 1 min

Max: 1 min

Stability

Refrigerate before use

Administration Notes

Used for hepatorenal syndrome and variceal bleeding.

Naloxone

Standard Diluent

NS

Final Concentration

0.4 mg/mL

Infusion Rate

IV push or infusion (0.4 - 4 mg/hr)

Max: Titrate to resp rate

Stability

24 hours

Administration Notes

Half life is short (30-60 mins). Rebound opioid toxicity common.

Protamine

Standard Diluent

Undiluted

Final Concentration

10 mg/mL

Infusion Rate

Give over 10 mins (Max 5 mg/min)

Max: 5 mg/min

Stability

Room temp

Administration Notes

Heparin reversal. Rapid push causes profound hypotension and bradycardia.

N-acetylcysteine

Standard Diluent

D5W

Final Concentration

Varies (3 bag regimen)

Infusion Rate

150mg/kg over 1hr, 50mg/kg over 4hr, 100mg/kg over 16hr

Max: Per protocol

Stability

24 hours

Administration Notes

Acetaminophen antidote. Anaphylactoid reactions common with first bag.

Fomepizole

Standard Diluent

NS or D5W (100 mL)

Final Concentration

15 mg/mL

Infusion Rate

Give over 30 mins

Max: 30 mins

Stability

24 hours

Administration Notes

Antidote for ethylene glycol / methanol poisoning.

Physostigmine

Standard Diluent

Undiluted

Final Concentration

1 mg/mL

Infusion Rate

Give over 5 mins (Max 1 mg/min)

Max: 1 mg/min

Stability

Room temp

Administration Notes

Antidote for anticholinergic toxicity. Have atropine ready for bradycardia.

Dexrazoxane

Standard Diluent

LR

Final Concentration

10 mg/mL

Infusion Rate

Give over 15 mins

Max: 15 mins

Stability

Use within 6 hours

Administration Notes

Antidote for anthracycline (doxorubicin) extravasation or cardiotoxicity.

Doxorubicin

Standard Diluent

NS

Final Concentration

2 mg/mL

Infusion Rate

IV Push over 3-5 mins

Max: 5 mins

Stability

Protect from light

Administration Notes

Severe vesicant. Highly cardiotoxic (lifetime dose limit).

Cisplatin

Standard Diluent

NS

Final Concentration

0.5 - 2 mg/mL

Infusion Rate

Over 1-2 hours

Max: Varies

Stability

Do NOT refrigerate

Administration Notes

Highly nephrotoxic and highly emetogenic.

Carboplatin

Standard Diluent

D5W or NS

Final Concentration

0.5 - 10 mg/mL

Infusion Rate

Over 15-60 mins

Max: 60 mins

Stability

24 hours

Administration Notes

Dosed via Calvert formula (based on AUC and GFR).

Paclitaxel

Standard Diluent

NS

Final Concentration

0.3 - 1.2 mg/mL

Infusion Rate

Over 3 hours

Max: 3 hours

Stability

27 hours (room temp)

Administration Notes

Requires non-PVC tubing and in-line filter. Premedicate for hypersensitivity.

Docetaxel

Standard Diluent

NS or D5W

Final Concentration

0.3 - 0.74 mg/mL

Infusion Rate

Over 1 hour

Max: 1 hour

Stability

4 hours

Administration Notes

Fluid retention is common; premedicate with dexamethasone.

Fluorouracil

Standard Diluent

NS or D5W

Final Concentration

Up to 50 mg/mL

Infusion Rate

Continuous infusion over 46-96 hours

Max: Varies

Stability

24 hours

Administration Notes

Can cause severe hand-foot syndrome.

Cyclophosphamide

Standard Diluent

NS

Final Concentration

20 mg/mL

Infusion Rate

Over 30-60 mins

Max: 60 mins

Stability

24 hours

Administration Notes

Risk of hemorrhagic cystitis (hydrate aggressively, sometimes use Mesna).

Ifosfamide

Standard Diluent

NS or D5W

Final Concentration

10 - 40 mg/mL

Infusion Rate

Over 2-24 hours

Max: Varies

Stability

24 hours

Administration Notes

High risk of hemorrhagic cystitis; ALWAYS give with Mesna.

Etoposide

Standard Diluent

NS

Final Concentration

0.2 - 0.4 mg/mL

Infusion Rate

Over 30-60 mins

Max: 60 mins

Stability

Concentration dependent (cracks if >0.4 mg/mL)

Administration Notes

Hypotension if infused too rapidly.

Vincristine

Standard Diluent

NS

Final Concentration

1 mg/mL

Infusion Rate

IV Push over 1 min

Max: 1 min

Stability

Refrigerate

Administration Notes

FATAL if given intrathecally. Severe vesicant.

Infliximab

Standard Diluent

NS only

Final Concentration

0.4 - 4 mg/mL

Infusion Rate

Over 2 hours

Max: 2 hours

Stability

24 hours (do not shake)

Administration Notes

Use in-line filter. High risk of infusion reactions.

Rituximab

Standard Diluent

NS or D5W

Final Concentration

1 - 4 mg/mL

Infusion Rate

Start at 50 mg/hr, titrate up

Max: 400 mg/hr

Stability

24 hours

Administration Notes

Premedicate with APAP and diphenhydramine.

Trastuzumab

Standard Diluent

NS only

Final Concentration

21 mg/mL

Infusion Rate

Over 30-90 mins

Max: 90 mins

Stability

28 days refrigerated

Administration Notes

Cardiotoxic (monitor LVEF). Do not mix with D5W.

Bevacizumab

Standard Diluent

NS

Final Concentration

1.4 - 16.5 mg/mL

Infusion Rate

Over 30-90 mins

Max: 90 mins

Stability

24 hours

Administration Notes

Risk of severe bleeding, GI perforation, and impaired wound healing.

Pembrolizumab

Standard Diluent

NS or D5W

Final Concentration

1 - 10 mg/mL

Infusion Rate

Over 30 mins

Max: 30 mins

Stability

24 hours refrigerated

Administration Notes

Immune-mediated adverse effects (pneumonitis, colitis, endocrinopathies).

Nivolumab

Standard Diluent

NS or D5W

Final Concentration

1 - 10 mg/mL

Infusion Rate

Over 30 mins

Max: 30 mins

Stability

24 hours

Administration Notes

Immune checkpoint inhibitor. Monitor for immune-mediated toxicities.

Tacrolimus

Standard Diluent

NS or D5W

Final Concentration

0.004 - 0.02 mg/mL

Infusion Rate

Continuous infusion

Max: Varies

Stability

24 hours

Administration Notes

Use non-PVC tubing. Highly nephrotoxic.

Cyclosporine

Standard Diluent

NS or D5W

Final Concentration

0.5 - 2.5 mg/mL

Infusion Rate

Over 2-6 hours

Max: 6 hours

Stability

24 hours

Administration Notes

Risk of anaphylaxis (cremophor vehicle). Premedicate.

Mycophenolate

Standard Diluent

D5W only

Final Concentration

6 mg/mL

Infusion Rate

Over 2 hours

Max: 2 hours

Stability

Use within 4 hours of reconstitution

Administration Notes

Do not mix or administer with other IV medications.

Basiliximab

Standard Diluent

NS or D5W

Final Concentration

0.4 mg/mL

Infusion Rate

Over 20-30 mins

Max: 30 mins

Stability

24 hours refrigerated

Administration Notes

Used for induction therapy in solid organ transplants.

Levetiracetam

Standard Diluent

NS or D5W

Final Concentration

5 - 15 mg/mL

Infusion Rate

Over 15 mins

Max: 15 mins

Stability

24 hours

Administration Notes

Can cause behavioral changes or agitation.

Fosphenytoin

Standard Diluent

NS or D5W

Final Concentration

1.5 - 25 mg PE/mL

Infusion Rate

Up to 150 mg PE/min

Max: 150 mg PE/min

Stability

24 hours

Administration Notes

Prodrug of phenytoin. Less risk of purple glove syndrome.

Phenytoin

Standard Diluent

NS only

Final Concentration

Max 5 mg/mL

Infusion Rate

Max 50 mg/min

Max: 50 mg/min

Stability

Use immediately

Administration Notes

Must use in-line filter. High risk of phlebitis/tissue necrosis.

Valproic Acid

Standard Diluent

NS or D5W

Final Concentration

Max 5 mg/mL

Infusion Rate

Over 60 mins (max 20 mg/min)

Max: 20 mg/min

Stability

24 hours

Administration Notes

Risk of hyperammonemia and hepatotoxicity.

Lacosamide

Standard Diluent

NS or D5W

Final Concentration

Max 10 mg/mL

Infusion Rate

Over 15-60 mins

Max: 60 mins

Stability

24 hours

Administration Notes

Can prolong PR interval (risk of heart block).

Brivaracetam

Standard Diluent

NS or D5W

Final Concentration

Max 5 mg/mL

Infusion Rate

IV Push over 2 mins or infusion

Max: 2 mins

Stability

24 hours

Administration Notes

Similar to levetiracetam but faster onset.

Palonosetron

Standard Diluent

Ready to use

Final Concentration

0.05 mg/mL

Infusion Rate

IV Push over 30 seconds

Max: 30 seconds

Stability

Room temp

Administration Notes

Long-acting 5-HT3 antagonist (half-life 40 hours).

Granisetron

Standard Diluent

NS or D5W

Final Concentration

0.02 - 0.2 mg/mL

Infusion Rate

IV Push over 30 seconds

Max: 30 seconds

Stability

24 hours

Administration Notes

Alternative to ondansetron; less QTc prolongation risk.

Fosaprepitant

Standard Diluent

NS

Final Concentration

1 mg/mL

Infusion Rate

Over 20-30 mins

Max: 30 mins

Stability

24 hours

Administration Notes

NK1 receptor antagonist for highly emetogenic chemo.

Famotidine

Standard Diluent

NS or D5W

Final Concentration

2 mg/mL

Infusion Rate

IV Push over 2 mins

Max: 2 mins

Stability

48 hours

Administration Notes

H2 blocker. Adjust dose in renal impairment.

Esomeprazole

Standard Diluent

NS or D5W

Final Concentration

0.8 mg/mL

Infusion Rate

Continuous infusion (8 mg/hr)

Max: 8 mg/hr

Stability

12 hours (protect from light)

Administration Notes

PPI used for acute upper GI bleeding.

Chlorpromazine

Standard Diluent

NS

Final Concentration

1 mg/mL

Infusion Rate

1 mg/min

Max: 1 mg/min

Stability

Protect from light

Administration Notes

High risk of severe hypotension when given IV.

Ibutilide

Standard Diluent

NS or D5W

Final Concentration

0.017 mg/mL

Infusion Rate

Over 10 mins

Max: 10 mins

Stability

24 hours

Administration Notes

Class III antiarrhythmic. High risk of Torsades (monitor ECG for 4 hrs).

Sotalol

Standard Diluent

NS or D5W

Final Concentration

1 - 2 mg/mL

Infusion Rate

Over 5 hours

Max: 5 hours

Stability

24 hours

Administration Notes

Initiation requires continuous ECG monitoring (QTc prolongation).

Metoprolol

Standard Diluent

Undiluted

Final Concentration

1 mg/mL

Infusion Rate

IV Push: 5 mg over 2 mins

Max: 3 doses max

Stability

Immediate use

Administration Notes

Cardioselective beta blocker.

Propranolol

Standard Diluent

NS or D5W

Final Concentration

1 mg/mL

Infusion Rate

IV Push: 1 mg over 1 min

Max: 1 min

Stability

24 hours

Administration Notes

Non-selective beta blocker. Used for thyroid storm.

Chlorothiazide

Standard Diluent

NS or D5W

Final Concentration

10 mg/mL

Infusion Rate

IV Push over 3-5 mins

Max: 5 mins

Stability

24 hours

Administration Notes

The only IV thiazide diuretic available.

Acetazolamide

Standard Diluent

Sterile Water

Final Concentration

50 mg/mL

Infusion Rate

IV Push over 1-2 mins

Max: 2 mins

Stability

12 hours

Administration Notes

Carbonic anhydrase inhibitor. Used for metabolic alkalosis or high ICP.

Torsemide

Standard Diluent

Undiluted

Final Concentration

10 mg/mL

Infusion Rate

IV Push over 2 mins

Max: 2 mins

Stability

24 hours

Administration Notes

Loop diuretic. Longer half-life than furosemide.

Ethacrynic Acid

Standard Diluent

D5W or NS

Final Concentration

1 mg/mL

Infusion Rate

Over 20-30 mins

Max: 30 mins

Stability

24 hours

Administration Notes

Used in patients with severe sulfa allergies.

Calcium Gluconate

Standard Diluent

NS or D5W

Final Concentration

10 - 50 mg/mL

Infusion Rate

1-2 g over 30-60 mins

Max: 60 mins

Stability

24 hours

Administration Notes

Can be given peripherally. Max rate 200 mg/min for cardiac arrest.

Calcium Chloride

Standard Diluent

NS or D5W

Final Concentration

100 mg/mL

Infusion Rate

IV Push (Code) or over 60 mins

Max: Varies

Stability

24 hours

Administration Notes

Requires central line (severe vesicant). 3x more potent than gluconate.

Potassium Chloride

Standard Diluent

NS (Avoid D5W)

Final Concentration

Max 10 mEq/100 mL peripheral

Infusion Rate

10 mEq/hr (Peripheral) or 20 mEq/hr (Central)

Max: 20 mEq/hr

Stability

24 hours

Administration Notes

NEVER give IV push. Fatal if given rapidly.

Sodium Bicarbonate

Standard Diluent

D5W or NS

Final Concentration

0.5 - 1 mEq/mL

Infusion Rate

IV Push (Arrest) or continuous infusion

Max: Varies

Stability

24 hours

Administration Notes

Highly alkaline. Ensure line patency.

Sodium Chloride 3% (Hypertonic)

Standard Diluent

Undiluted

Final Concentration

3%

Infusion Rate

Varies (e.g. 30 mL/hr)

Max: Varies

Stability

24 hours

Administration Notes

Must be given via central line. Risk of osmotic demyelination if corrected too fast.

Thiamine

Standard Diluent

NS or D5W

Final Concentration

1 - 10 mg/mL

Infusion Rate

Over 15-30 mins

Max: 30 mins

Stability

24 hours

Administration Notes

Give BEFORE glucose in malnourished/alcoholic patients to prevent Wernicke's encephalopathy.

Folic Acid

Standard Diluent

NS or D5W

Final Concentration

Varies

Infusion Rate

IV Push or short infusion

Max: Varies

Stability

24 hours

Administration Notes

Usually given with thiamine in a 'banana bag'.

Cyanocobalamin

Standard Diluent

NS or D5W

Final Concentration

Varies

Infusion Rate

IM preferred, can be given IV

Max: Varies

Stability

Protect from light

Administration Notes

Vitamin B12. Can cause hypokalemia as RBCs rapidly form.

Dexmedetomidine

Standard Diluent

NS

Final Concentration

4 mcg/mL

Infusion Rate

0.2 - 1.5 mcg/kg/hr

Max: 1.5 mcg/kg/hr

Stability

24 hours

Administration Notes

Does not cause respiratory depression. Watch for bradycardia and hypotension.

Isoproterenol

Standard Diluent

D5W

Final Concentration

4 mcg/mL

Infusion Rate

2 - 10 mcg/min

Max: Titrate to HR

Stability

24 hours

Administration Notes

Pure beta agonist. Refractory bradycardia.